巴氯芬 分析标准品
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| 包装规格: | 25mg in glass bottle |
| 产品描述: | γ-氨基丁酸(GABA)的亲脂性衍生物,一种口服有效,选择性的代谢型GABA-B受体(GABABR)激动剂。Baclofen具有高的血脑屏障渗透率。Baclofen有用于肌肉痉挛研究的潜力。 Baclofen is a GABA agonist specific for GABA-B receptors. Baclofen is a synthetic chlorophenyl-butanoic acid derivative used to treat spasms due to spinal cord damage and multiple sclerosis, muscle-relaxing. It acts at spinal and supraspinal sites, reducing excitatory transmission. |
| 保存条件: | 室温 |
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