[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
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| 包装规格: | 1mg 5mg in glass bottle |
| 产品简介: | 一种有效的,选择性神经肽 YY5 受体激动剂。 |
| 溶解性: | DMSO :100 mg/mL(23.77 mM;超声助溶) |
| 储备液保存: | -80°C, 6 months -20°C, 1 month (sealed storage, away from moisture) |
| 靶点: | hY5 receptor:0.24 nM (IC50);hY1 receptor:530 nM (IC50);hY2 receptor:>500 nM (IC50);hY4 receptor:51 nM (IC50) |
| 体外研究: | [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide has IC50s of 530 nM, >500 nM, 51 nM for binding to the hY1, hY4, hY2 receptors. |
| 体内研究: | [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide (0.2, 2 nmol/rat) induces a high amount of food intake in a dose-dependent manner in adult male rats weighing 340-400 g. |
| 保存条件: | -20℃ |
| 注意事项: | 1、为了您的安全和健康,请穿实验服并戴一次性手套操作。 2、以上信息仅做参考交流之用。 |
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