盐酸西维美林 ≥98%
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| 包装规格: | 1mg 5mg 10mg 25mg 50mg 100mg in glass bottle |
| 产品简介: | 一种乙酰胆碱的奎尼丁衍生物,也是一种选择性的和口服活性的毒蕈碱型 M1和M3 受体激动剂。Cevimeline hydrochloride 可刺激唾液腺分泌,并可用作口干症的一种催涎剂。Cevimeline hydrochloride 可穿过血脑屏障。 |
| 溶解性: | 溶于水(≥50mg/mL) |
| 储备液保存: | -80°C, 6 months -20°C, 1 month (sealed storage, away from moisture) |
| 靶点: | Muscarinic M1 and M3 receptor |
| 体外研究: | In digested parotid cells, Cevimeline (0.1-100 μM) increases the intracellular Ca2+ concentration. |
| 体内研究: | Cevimeline (0.008-0.016 mg/kg; intraperitoneal injection; male Wistar rats) treatment shows slowly increasing and lasting salivation, and increased blood flow increment in the parotid gland and pressor response. Cevimeline inhibits angiotensin II-induced water intake and neuronal activity in the subfornical organ at 0.016 mg/kg. |
| 保存条件: | -20℃ |
| 注意事项: | 1、为了您的安全和健康,请穿实验服并戴一次性手套操作。 2、以上信息仅做参考交流之用。 |
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