Gemfibrozil 促销  ≥98%

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包装规格:25g 100g 500g in poly bottle
产品简介:一种PPAR-α激活剂,是一种降脂药;Gemfibrozil同时是P450的非选择性抑制剂,对CYP2C9,2C19,2C8和1A2的Ki值分别为5.8,24,69和82μM。 Gemfibrozil is a peroxisome proliferator receptor alpha agonist. The mechanism of action of gemfibrozil is as a Peroxisome Proliferator-activated Receptor alpha Agonist. The chemical classification of gemfibrozil is PPAR alpha. Gemfibrozil is a lipid-regulating agent that lowers elevated serum lipids primarily by decreasing serum triglycerides with a variable reduction in total cholesterol.
溶解性:溶于DMSO(100mg/ml超声)
产品描述:一种PPAR-α激活剂,是一种降脂药;Gemfibrozil同时是P450的非选择性抑制剂,对CYP2C9,2C19,2C8和1A2的Ki值分别为5.8,24,69和82μM。Gemfibrozil is a peroxisome proliferator receptor alpha agonist. The mechanism of action of gemfibrozil is as a Peroxisome Proliferator-activated Receptor alpha Agonist. The chemical classification of gemfibrozil is PPAR alpha. Gemfibrozil is a lipid-regulating agent that lowers elevated serum lipids primarily by decreasing serum triglycerides with a variable reduction in total cholesterol.
保存条件:室温